Development of β-carboline-benzothiazole hybrids via carboxamide formation as cytotoxic agents: DNA intercalative topoisomerase IIα inhibition and apoptosis induction

Author:

Tokala Ramya,Mahajan Surbhi,Kiranmai Gaddam,Sigalapalli Dilep Kumar,Sana Sravani,John Stephy Elza,Nagesh Narayana,Shankaraiah Nagula

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference65 articles.

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2. Discovery of novel topoisomerase II inhibitors by medicinal chemistry approaches;Hu;J. Med. Chem.,2018

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4. Therapeutic intervention by the simultaneous inhibition of DNA repair and type I or type II DNA topoisomerases: one strategy, many outcomes;Wesierska-Gadek;Future Med. Chem.,2012

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