Identification of 2(1H)-pyrimidinones as potential EGFR T790M inhibitors for the treatment of gefitinib-resistant non-small cell lung cancer-Reference-Cited by-同舟云学术

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Identification of 2(1H)-pyrimidinones as potential EGFR T790M inhibitors for the treatment of gefitinib-resistant non-small cell lung cancer

Published:2019-08 Issue: Volume:89 Page:102994
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Huang Jianping,Huang Jiaxin,Wang Ning,Wang Luhong,Li Lei,Wang Changyuan,Sun Xiuli,Li Yongming,Huang Guoping,Ma Xiaodong

Funder

National Natural Science Foundation of China

Research Fund of Higher Education of Liaoning province

National Natural Science Foundation of Liaoning province

Cultivation Project of Youth Techstars, Dalian, China

Natural Science Foundation of Science and Technology Department of Jiangxi Province

Natural Science Foundation of Education Department of Jiangxi Province

Natural Science Foundation of Nanchang City

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference23 articles.

1. Non-small cell lung cancer: epidemiology, risk factors, treatment, and survivorship;Molina;Mayo. Clin. Proc.,2008

2. Epidermal growth factor receptor mutations in lung cancer;Sharma;Nat. Rev. Cancer,2007

3. Gefitinib (Iressa): a novel treatment for non-small cell lung cancer;Vansteenkiste;Expert. Rev. Anticancer. Ther.,2004

4. Erlotinib: a new therapeutic approach for non-small cell lung cancer;Bonomi;Expert. Opin. Investig. Drugs.,2003

5. Challenges and perspectives on the development of small-molecule EGFR inhibitors against T790M-mediated resistance in non-small-cell lung cancer;Song;J. Med. Chem.,2016

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1. Structural Perspectives in the Development of Novel EGFR Inhibitors for the Treatment of NSCLC;Mini-Reviews in Medicinal Chemistry;2024-10

2. Design and synthesis of novel uracil-linked Schiff bases as dual histone deacetylase type II/topoisomerase type I inhibitors with apoptotic potential;Future Medicinal Chemistry;2023-06

3. Design, synthesis and biological evaluation of novel 3,4-dihydro-2H-[1,4]oxazino [2,3-f]quinazolin derivatives as EGFR-TKIs;Bioorganic & Medicinal Chemistry Letters;2023-01

4. Overview of the multifaceted resistances toward EGFR-TKIs and new chemotherapeutic strategies in non-small cell lung cancer;Biochemical Pharmacology;2022-11

5. Comparative experimental and DFT analysis of novel indole tagged [1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one hybrid;Journal of Molecular Structure;2022-09

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