Synthesis, molecular docking and biological evaluation of 2-(thiophen-2-yl)-1H-indoles as potent HIV-1 non-nucleoside reverse transcriptase inhibitors-Reference-Cited by-同舟云学术

Synthesis, molecular docking and biological evaluation of 2-(thiophen-2-yl)-1H-indoles as potent HIV-1 non-nucleoside reverse transcriptase inhibitors

Published:2020-01 Issue: Volume:95 Page:103521
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

El-Hussieny Marwa,El-Sayed Naglaa F.,Ewies Ewies F.,Ibrahim Nabila M.,Mahran Mohamed R.H.,Fouad Marwa A.

Funder

National Research Centre, Egypt

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

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5. Phenethylthiazolethiourea (PETT), compounds, a new class of HIV-1 reverse transcriptase inhibitors. 1. Synthesis and basic structure-activity relationship studies of PETT analogs;Bell;J. Med. Chem.,1995

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