Syntheses and studies of deuterated Imdiazo[1,2-a]pyridine-3-carboxamides with potent anti-tuberculosis activity and improved metabolic properties-Reference-Cited by-同舟云学术

Syntheses and studies of deuterated Imdiazo[1,2-a]pyridine-3-carboxamides with potent anti-tuberculosis activity and improved metabolic properties

Published:2022-11 Issue: Volume:128 Page:106074
ISSN:0045-2068
Container-title:Bioorganic Chemistry
language:en
Short-container-title:Bioorganic Chemistry

Author:

Liu Rui,Marshall Kate,Ma Rui,Lien Thi Pham Kim,Shetye Gauri,Liu Zhihao,Cho Sanghyun,Jeong Hyunyoung,Franzblau Scott G.,Moraski Garrett C.,Miller Marvin J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference38 articles.

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4. (a) Moraski, G. C.; Markley, L. D.; Cramer, J.; Hipskind, P. A.; Boshoff, H.; Bailey, M.; Alling, T.; Ollinger, J.; Parish, T.; Miller, M. J. Advancement of Imidazo[1,2-a]pyridines with Improved Pharmacokinetics and Nanomolar Activity AgainstMycobacterium tuberculosis ACS Med. Chem. Lett., 2013, 4, 675-679. doi: 10.1021/ml400088y. (b) Ollinger, J.; Bailey, M. A.; Moraski, G. C.; Casey, A.; Florio, S.; Alling, T.; Miller, M. J.; Parish, T. A Dual Read-Out Assay to Evaluate the Potency of Compounds Active againstMycobacterium tuberculosis. PLOS ONE 8(4): e60531.https://doi.org/10.1371/journal.pone.0060531. (c) Moraski, G. C.; Miller, P. A.; Bailey, M. A.; Ollinger, J.; Parish, T.; Boshoff, H. I.; Cho, S.; Anderson, J. R.; Mulugeta, S.; Franzblau, S. G.; Miller, M. J. Putting Tuberculosis (TB) To Rest: Transformation of the Sleep Aid, Ambien, and “Anagrams” Generated Potent Antituberculosis Agents ACS Inf. Dis., 2015, 1, 85-90. https://doi.org/10.1021/id500008t. (d) Moraski, G. C.; Bristol, R.; Seeger, N.; Boshoff, H. I.; Tsang, P. S.; Miller, M. J. Preparation and Evaluation of Potent Pentafluorosulfanyl-Substituted Anti-Tuberculosis Compounds, ChemMedChem., 2017, 12, 1108-1115. https://doi.org/10.1002/cmdc.201700170.

5. Scaffold-switching: An exploration of 5,6-fused bicyclic heteroaromatics systems to afford antituberculosis activity akin to the imidazo[1,2-a]pyridine-3-carboxylates;Moraski;Bioorg. Med. Chem. Lett.,2014

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