Design, synthesis, and molecular docking of novel pyrazole-chalcone analogs of lonazolac as 5-LOX, iNOS and tubulin polymerization inhibitors with potential anticancer and anti-inflammatory activities
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry
Reference67 articles.
1. Imidazoles as potential anticancer agents;Ali;Medchemcomm,2017
2. Molecular targets and anticancer activity of quinoline–chalcone hybrids: literature review;Mohamed;RSC Adv.,2020
3. Discovery of new quinoxaline-2(1H)-one-based anticancer agents targeting VEGFR-2 as inhibitors: Design, synthesis, and anti-proliferative evaluation;El-Adl;Bioorg. Chem.,2021
4. Design, synthesis and biological evaluation of (E)-2-(2-arylhydrazinyl)quinoxalines, a promising and potent new class of anticancer agents;Rodrigues;Bioorg. Med. Chem. Lett.,2014
5. Utilization of cyanopyridine in design and synthesis of first-in-class anticancer dual acting PIM-1 kinase/HDAC inhibitors;Bass;Bioorg. Chem.,2022
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