1,2,3-triazole tethered Indole-3-glyoxamide derivatives as multiple inhibitors of 5-LOX, COX-2 & tubulin: Their anti-proliferative & anti-inflammatory activity
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry
Reference34 articles.
1. The fractions of cancer attributable to modifiable factors: a global review;Whiteman;Cancer Epidemiol.,2016
2. Antimitotic agents of natural origin;Nagle;Curr. Drug Target.,2006
3. Microtubule inhibitors: differentiating tubulin-inhibiting agents based on mechanisms of action, clinical activity, and resistance;Perez;Mol. Cancer Ther.,2009
4. Drugs that target dynamic microtubules: a new molecular perspective;Stanton;Med. Res. Rev.,2011
5. Licofelone, a dual COX/5-LOX inhibitor, induces apoptosis in HCA-7 colon cancer cells through the mitochondrial pathway independently from its ability to affect the arachidonic acid cascade;Simona;Carcinogenesis,2008
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