Discovery of novel phenyl triazole analogs as TRK/ALK dual inhibitors with prospective antitumor effects
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry
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4. A next-Generation TRK kinase inhibitor overcomes acquired resistance to prior TRK kinase inhibition in patients with TRK fusion-positive solid tumors;Drilon;Cancer Discovery.,2017
5. TPX-0005, a novel ALK/ROS1/TRK inhibitor effectively inhibited a broad spectrum of mutations including solvent front ALKG1202R, ROS1G2032R and TRKAG595R mutants;Cui;Eur. J. Cancer,2016
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1. Anaplastic lymphoma kinase inhibitors—a review of anticancer properties, clinical efficacy, and resistance mechanisms;Frontiers in Pharmacology;2023-10-25
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