Imidazo[1,2-a]quinazolines as novel, potent EGFR-TK inhibitors: Design, synthesis, bioactivity evaluation, and in silico studies

Author:

Hasanvand Zaman,Oghabi Bakhshaiesh Tayebeh,Peytam Fariba,Firoozpour Loghman,Hosseinzadeh Elaheh,Motahari Rasoul,Moghimi Setareh,Nazeri Elaheh,Toolabi Mahsa,Momeni Farhad,Bijanzadeh Hamidreza,Khalaj Ali,Baratte Blandine,Josselin Béatrice,Robert Thomas,Bach Stéphane,Esmaeili Rezvan,Foroumadi AlirezaORCID

Funder

Tehran University of Medical Sciences and Health Services

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference54 articles.

1. WebMD, https://www.who.int/news-room/fact-sheets/detail/cancer.

2. Current molecular-targeted therapies in NSCLC and their mechanism of resistance;Schrank;Cancers,2018

3. An overview of cancer treatments;Anderson;Pharm. J.,2009

4. The Aurora kinase inhibitors in cancer research and therapy;Cicenas;J. Cancer Res. Clin. Oncol.,2016

5. Properties of FDA-approved small molecule protein kinase inhibitors: a update;Roskoski;Pharmacol. Res.,2021

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