Pharmacokinetics and safety of rilpivirine in healthy Japanese subjects and exploration of ethnic sensitivity of rilpivirine pharmacokinetics with physiologically based pharmacokinetic model approach

Author:

Ohta Kentaro,Matsushima Nobuko,Tanii Hiromi,Crauwels Herta,Kudo Toshiyuki,Ito Kiyomi

Publisher

Elsevier BV

Subject

Pharmacology (medical),Pharmaceutical Science,Pharmacology

Reference24 articles.

1. TMC278, a next-generation nonnucleoside reverse transcriptase inhibitor (NNRTI), active against wild-type and NNRTI-resistant HIV-1;Azijn;Antimicrob Agents Chemother,2010

2. REKAMBYS® (rilpivirine) [prescribing information]. Janssen-Cilag International NV. Beerse, Belgium.

3. CABENUVA® (cabotegravir extended release injectable suspension; rilpivirine extended-release injectable suspension) [prescribing information]. ViiV Healthcare, NC, USA.

4. Rilpivirine

5. Application of approval for manufacturing or importing anti-HIV drugs,1998

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