14β-Chlorocinnamoylamino derivatives of metopon: long-term μ-opioid receptor antagonists

Author:

McLaughlin Jay P,Sebastian Alice,Archer Sydney,Bidlack Jean M

Publisher

Elsevier BV

Subject

Pharmacology

Reference42 articles.

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2. Archer, S., A. Seyed-Mozaffari, Q. Jiang and J.M. Bidlack, 1994, 14α,14′β-[Dithiobis[2-oxo-2,1-ethanediyl)imino]]bis[(7,8-dihydromorphinone) and 14α,14′β-[dithiobis[2-oxo-2,1-ethanediyl)imino]]bis[7,8-dihydro-N-(cyclopropylmethyl)normorphinone]: chemistry and opioid binding properties, J. Med. Chem. 37, 1578.

3. Bidlack, J.M, D.K. Frey, R.K. Kaplan, A. Seyed-Mozaffari and S. Archer, 1990, Affinity labeling of μ opioid receptors by sulfhydryl alkylating derivatives of morphine and morphinone, Mol. Pharmacol. 37, 50.

4. Bidlack, J.M., R.A. Kaplan, R.A. Subbramanian, A. Seyed-Mozaffari and S. Archer, 1993, Affinity labeling of the μ opioid receptor in bovine striatal membranes with [3H]-14-β-(bromoacetamido)-7,8-dihydromorphine, Biochemistry 32, 6703.

5. Bradford, M.M., 1976, A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding, Anal. Biochem. 72, 248.

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