The assessment of antagonist potency under conditions of transient response kinetics-Reference-Cited by-同舟云学术

The assessment of antagonist potency under conditions of transient response kinetics

Published:1999-10 Issue:3 Volume:382 Page:217-227
ISSN:0014-2999
Container-title:European Journal of Pharmacology
language:en
Short-container-title:European Journal of Pharmacology

Author:

Christopoulos Arthur,Parsons Ann M.,Lew Michael J.,El-Fakahany Esam E.

Publisher

Elsevier BV

Subject

Pharmacology

Reference30 articles.

1. Some quantitative uses of drug antagonists;Arunlakshana;Br. J. Pharmacol.,1959

2. Operational models of pharmacological agonism;Black;Proc. R. Soc. (London) B,1983

3. Unsurmountable antagonism to 5-hydroxytryptamine in rat kidney results from pseudoirreversible inhibition rather than multiple receptors or allosteric receptor modulation;Bond;J. Pharmacol. Exp. Ther.,1989

4. Promiscuous or heterogeneous muscarinic receptors in rat atria? II. Antagonism of responses to carbachol by pirenzepine;Boselli;Eur. J. Pharmacol.,1990

5. Muscarinic receptors — characterization, coupling and function;Caulfield;Pharmacol. Ther.,1993

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