The preparation and sar of 4-(anilino), 4-(phenoxy), and 4-(thiophenoxy)-quinazolines: Inhibitors of p56lck and EGF-R tyrosine kinase activity-Reference-Cited by-同舟云学术

The preparation and sar of 4-(anilino), 4-(phenoxy), and 4-(thiophenoxy)-quinazolines: Inhibitors of p56lck and EGF-R tyrosine kinase activity

Published:1997-02 Issue:4 Volume:7 Page:417-420
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Myers Michael R.,Setzer Natalie N.,Spada Alfred.P.,Zulli Allison L.,Hsu Chin-Yi J.,Zilberstein Asher,Johnson Susan E.,Hook Linda E.,Jacoski Mary V.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference28 articles.

1. Partially disclosed in Myers, M. R.; Spada, A. P.; Maguire, M. P.; Persons, P. E.; Zilberstein, A., Hsu, C.-Y.; Johnson, S., WO PCT Appl. 95/15758, 1995.

2. The Src family of tyrosine protein kinases in hemopoietic signal transduction

3. Transmembrane Signaling of T Lymphocytes by Ligand-Induced Receptor Complex Assembly

4. T cell antigen receptor activation pathways: The tyrosine kinase connection

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