Bioisosteres of 9-Carboxymethyl-4-oxo-imidazo[1,2- a ]indeno[1,2- e ]pyrazin-2-carboxylic acid derivatives. Progress towards selective, potent In Vivo AMPA antagonists with longer durations of action-Reference-Cited by-同舟云学术

Bioisosteres of 9-Carboxymethyl-4-oxo-imidazo[1,2- a ]indeno[1,2- e ]pyrazin-2-carboxylic acid derivatives. Progress towards selective, potent In Vivo AMPA antagonists with longer durations of action

Published:2001-01 Issue:2 Volume:11 Page:127-132
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Jimonet Patrick,Bohme Georg Andrees,Bouquerel Jean,Boireau Alain,Damour Dominique,Debono Marc Williams,Genevois-Borella Arielle,Hardy Jean-Claude,Hubert Philippe,Manfré Franco,Nemecek Patrick,Pratt Jeremy,Randle John C.R.,Ribeill Yves,Stutzmann Jean-Marie,Vuilhorgne Marc,Mignani Serge

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference40 articles.

1. Triggering and execution of neuronal death in brain ischaemia: two phases of glutamate release by different mechanisms

2. The Role of Excitotoxicity in Neurodegenerative Disease

3. Molecular Diversity of Glutamate Receptors and Implications for Brain Function

4. For a recent review, see: Nature 1999, 399(Suppl), and references cited therein.

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