Design, synthesis and In vitro evaluation of potent, novel, small molecule inhibitors of plasminogen activator inhibitor-1-Reference-Cited by-同舟云学术

Design, synthesis and In vitro evaluation of potent, novel, small molecule inhibitors of plasminogen activator inhibitor-1

Published:2002-04 Issue:7 Volume:12 Page:1063-1066
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Folkes Adrian,Brown S.David,Canne Lynne E.,Chan Jocelyn,Engelhardt Erin,Epshteyn Sergey,Faint Richard,Golec Julian,Hanel Art,Kearney Patrick,Leahy James W.,Mac Morrison,Matthews David,Prisbylla Michael P.,Sanderson Jason,Simon Reyna J.,Tesfai Zerom,Vicker Nigel,Wang Shouming,Webb Robert R.,Charlton Peter

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference18 articles.

1. The plasminogen activator/plasmin system.

2. Structure of plasminogen activator inhibitor 1 (PAI-1) and its function in fibrinolysis: an update

3. The serpin superfamily of proteinase inhibitors: structure, function, and regulation.

4. The status of PAI-1 as a risk factor for arterial and thrombotic disease: A review

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