Synthesis and Biological Evaluation of 2-Indolyloxazolines as a New Class of Tubulin Polymerization Inhibitors. Discovery of A-289099 as an Orally Active Antitumor Agent-Reference-Cited by-同舟云学术

Synthesis and Biological Evaluation of 2-Indolyloxazolines as a New Class of Tubulin Polymerization Inhibitors. Discovery of A-289099 as an Orally Active Antitumor Agent

Published:2002-02 Issue:3 Volume:12 Page:465-469
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Li Qun,Woods Keith W.,Claiborne Akiyo,Gwaltney, II Stephen L.,Barr Kenneth J.,Liu Gang,Gehrke Laura,Credo R.Bruce,Hui Yu Hua,Lee Jang,Warner Robert B.,Kovar Peter,Nukkala Michael A.,Zielinski Nicolette A.,Tahir Stephen K.,Fitzgerald Michael,Kim Ki H.,Marsh Kennan,Frost David,Ng Shi-Chung,Rosenberg Saul,Sham Hing L.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference21 articles.

1. Chapter 14. Antimitotic Agents

2. New inhibitors of tubulin polymerisation

3. Recent strategies in the development of taxane anticancer drugs

4. Taxanes and other microtubule stabilising agents

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