Synthesis of substituted 5[H]phenanthridin-6-ones as potent poly(ADP-ribose)polymerase-1 (PARP1) inhibitors

Author:

Li Jia-He,Serdyuk Larisa,Ferraris Dana V.,Xiao Ge,Tays Kevin L.,Kletzly Paul W.,Li Weixing,Lautar Susan,Zhang Jie,Kalish Vincent J.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference13 articles.

1. Poly(ADP-ribose) Polymerase-1 in the Nervous System

2. Zhang, J. In Emerging Drugs: The Prospect for Improved Medicines; Fitzgerald, J. D., Bowman, W. C., Taylor, J. B., Eds.; Ashley: London, 1999; Vol. 4, pp 209–221.

3. Li, J.-H.; Kalish, V. J.; Lautar, S.; Zhang, J. Abstract of Papers, Part 1, 220th National Meeting of the American Chemical Society, Washington, DC, Aug 2000, MEDI 154.

4. GPI 6150 Prevents H2O2 Cytotoxicity by Inhibiting Poly(ADP-ribose) Polymerase

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