Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 3: A proposed pharmacophore model for 1-[N-(methyl)-N-(phenylsulfonyl)amino]-2-(phenyl)-4-[4-(substituted)piperidin-1-yl]butanes-Reference-Cited by-同舟云学术

Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 3: A proposed pharmacophore model for 1-[N-(methyl)-N-(phenylsulfonyl)amino]-2-(phenyl)-4-[4-(substituted)piperidin-1-yl]butanes

Published:2001-09 Issue:18 Volume:11 Page:2469-2473
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Finke Paul E.,Meurer Laura C.,Oates Bryan,Shah Shrenik K.,Loebach Jennifer L.,Mills Sander G.,MacCoss Malcolm,Castonguay Laurie,Malkowitz Lorraine,Springer Martin S.,Gould Sandra L.,DeMartino Julie A.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference20 articles.

1. Human Chemokines: An Update

2. Host factors and the pathogenesis of HIV-induced disease

3. Homozygous Defect in HIV-1 Coreceptor Accounts for Resistance of Some Multiply-Exposed Individuals to HIV-1 Infection

4. The role of viral phenotype and CCR-5 gene defects in HIV-1 transmission and disease progression

5. HIV-1 entry – an expanding portal for drug discovery

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