Pharmacological, Pharmacokinetic, Pharmacodynamic and Physicochemical Characterization of FE 205030: A Potent, Fast Acting, Injectable CGRP Receptor Antagonist for the Treatment of Acute Episodic Migraine-Reference-Cited by-同舟云学术

Pharmacological, Pharmacokinetic, Pharmacodynamic and Physicochemical Characterization of FE 205030: A Potent, Fast Acting, Injectable CGRP Receptor Antagonist for the Treatment of Acute Episodic Migraine

Published:2022-01 Issue:1 Volume:111 Page:247-261
ISSN:0022-3549
Container-title:Journal of Pharmaceutical Sciences
language:en
Short-container-title:Journal of Pharmaceutical Sciences

Author:

Srinivasan Karthik,Kozminski Kirk,Zhang Ying,Wisniewski Kazimierz,Kohout Trudy,Wisniewska Halina,Harris Geoffrey,Lindstrom Beatriz,Hargrove Diane

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference32 articles.

1. Alternative RNA processing in calcitonin gene expression generates mRNAs encoding different polypeptide products;Amara;Nature,1982

2. Calcitonin gene-related peptide: physiology and pathophysiology;Russell;Physiol Rev,2014

3. Expression in brain of a messenger RNA encoding a novel neuropeptide homologous to calcitonin gene-related peptide;Amara;Science,1985

4. Isolation and characterization of human calcitonin gene-related peptide;Morris;Nature,1984

5. Distribution and chromatographic characterisation of CGRP-like immunoreactivity in the brain and gut of the rat;Mulderry;Regul Pept,1985

Cited by 5 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Examining the shared etiology of psychopathology with genome-wide association studies;Physiological Reviews;2023-04-01

2. CGRP physiology, pharmacology, and therapeutic targets: migraine and beyond;Physiological Reviews;2023-04-01

3. A systematic review with expert opinion on the role of gepants for the preventive and abortive treatment of migraine;Expert Review of Neurotherapeutics;2022-06-03

4. Lipidated Calcitonin Gene-Related Peptide (CGRP) Peptide Antagonists Retain CGRP Receptor Activity and Attenuate CGRP Action In Vivo;Frontiers in Pharmacology;2022-03-07

5. Novel Macrocyclic Antagonists of the Calcitonin Gene-Related Peptide Receptor: Design, Realization, and Structural Characterization of Protein–Ligand Complexes;ACS Chemical Neuroscience;2022-03-04