Auto-Induction of Intestinal First-Pass Effect Related Time-Dependent Pharmacokinetics of Artemisinin Rather than Dihydroartemisinin

Author:

Chai Liqing,Wang Rongrong,Wang Yan,Guo Wenju,Li Ning,Zuo Hengtong,Wang Yidan,Duan Danyu,Ren Guolian,Zheng Bin,Wang Ruili,Zhang ShuqiuORCID

Funder

National Natural Science Foundation of China

Shanxi Platform Base and Talent Special Project

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference28 articles.

1. Antimalarial Drug Combination Therapy. Report of a WHO Technical Consultation,2001

2. Evaluation of P450 inhibition and induction by artemisinin antimalarials in human liver microsomes and primary human hepatocytes;Xing;Drug Metab Dispos,2012

3. Pharmacokinetics of artemisinin-type compounds;Navaratnam;Clin Pharmacokinet,2000

4. Evidence for timedependent artemisinin kinetics in adults with uncomplicated malaria;Ashton;Pharm Pharmacol Lett,1996

5. Artemisinin pharmacokinetics is time-dependent during repeated oral administration in healthy male adults;Ashton;Drug Metab Dispos,1998

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