Allosteric binding sites at the receptor–lipid bilayer interface: novel targets for GPCR drug discovery
Author:
Funder
National Natural Science Foundation of China
Publisher
Elsevier BV
Subject
Drug Discovery,Pharmacology
Reference85 articles.
1. Subcellular organization of GPCR signaling;Eichel;Trends Pharmacol. Sci.,2018
2. GPCR dynamics: structures in motion;Latorraca;Chem. Rev.,2017
3. The G-protein-coupled receptors in the human genome form five main families. Phylogenetic analysis, paralogon groups, and fingerprints;Fredriksson;Mol. Pharmacol.,2003
4. The structure and function of G-protein-coupled receptors;Rosenbaum;Nature,2009
5. Diverse GPCRs exhibit conserved water networks for stabilization and activation;Venkatakrishnan;Proc. Natl. Acad. Sci. U. S. A.,2019
Cited by 42 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Designed dualsteric modulators: A novel route for drug discovery;Drug Discovery Today;2024-10
2. Exploring the constitutive activation mechanism of the class A orphan GPR20;Acta Pharmacologica Sinica;2024-09-10
3. Green Synthesis of Diphenyl‐Substituted Alcohols Via Radical Coupling of Aromatic Alcohols Under Transition‐Metal‐Free Conditions;ChemistryOpen;2024-08-22
4. Lipid Trolling to Optimize A3 Adenosine Receptor-Positive Allosteric Modulators (PAMs);Journal of Medicinal Chemistry;2024-07-03
5. Know your molecule: pharmacological characterization of drug candidates to enhance efficacy and reduce late-stage attrition;Nature Reviews Drug Discovery;2024-06-18
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3