Case study: adapting in vitro blood–brain barrier models for use in early-stage drug discovery

Author:

Vandenhaute Elodie,Sevin Emmanuel,Hallier-Vanuxeem Dorothée,Dehouck Marie-Pierre,Cecchelli Roméo

Publisher

Elsevier BV

Subject

Drug Discovery,Pharmacology

Reference30 articles.

1. Assessment of the blood-brain barrier in CNS drug discovery;Jeffrey;Neurobiol. Dis.,2010

2. Strategies to assess bloodbrain barrier penetration;Di;Expert Opin. Drug Discov.,2008

3. Distribution of morphine 6-glucuronide and morphine across the blood-brain barrier in awake, freely moving rats investigated by in vivo microdialysis sampling;Aasmundstad;J. Pharmacol. Exp. Ther.,1995

4. The effect of plasma protein binding on in vivo efficacy: misconceptions in drug discovery;Smith;Nat. Rev. Drug Discov.,2010

5. On the rate and extent of drug delivery to the brain;Hammarlund-Udenaes;Pharm. Res.,2008

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