Drugging specific conformational states of GPCRs: challenges and opportunities for computational chemistry
Author:
Funder
DFG
FEDER
Publisher
Elsevier BV
Subject
Drug Discovery,Pharmacology
Reference49 articles.
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2. Restructuring G-protein-coupled receptor activation;Audet;Cell,2012
3. Ligand-dependent perturbation of the conformational ensemble for the GPCR β2 adrenergic receptor revealed by HDX;West;Structure,2011
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5. Biased signaling pathways in β2-adrenergic receptor characterized by 19F-NMR;Liu;Science,2012
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