Synthesis and in vitro examination of [124I]-, [125I]- and [131I]-2-(4-iodophenylamino) pyrido[2,3-d]pyrimidin-7-one radiolabeled Abl kinase inhibitors

Author:

Veach Darren R.,Namavari Mohammad,Beresten Tatiana,Balatoni Julius,Minchenko Maria,Djaballah Hakim,Finn Ronald D.,Clarkson Bayard,Gelovani Juri G.,Bornmann William G.,Larson Steven M.

Publisher

Elsevier BV

Subject

Cancer Research,Radiology Nuclear Medicine and imaging,Molecular Medicine

Reference45 articles.

1. The pyrido[2,3-d]pyrimidine derivative PD180970 inhibits p210Bcr–Abl tyrosine kinase and induces apoptosis of K562 leukemic cells;Dorsey;Cancer Res,2000

2. Characterization of potent inhibitors of the Bcr–Abl and the c-kit receptor tyrosine kinases;Wisniewski;Cancer Res,2002

3. Biochemical and cellular effects of c-Src kinase-selective pyrido[2, 3-d]pyrimidine tyrosine kinase inhibitors;Kraker;Biochem Pharmacol,2000

4. The biology of chronic myeloid leukemia;Faderl;N Engl J Med,1999

5. The development of imatinib as a therapeutic agent for chronic myeloid leukemia;Deininger;Blood,2004

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