Stereoselective synthesis of chiral β-amino trifluoromethyl alcohol: development of a manufacturing process for a key intermediate in the production of a novel elastase inhibitor, AE-3763-Reference-Cited by-同舟云学术

Stereoselective synthesis of chiral β-amino trifluoromethyl alcohol: development of a manufacturing process for a key intermediate in the production of a novel elastase inhibitor, AE-3763

Published:2010-08 Issue:15 Volume:21 Page:1855-1860
ISSN:0957-4166
Container-title:Tetrahedron: Asymmetry
language:en
Short-container-title:Tetrahedron: Asymmetry

Author:

Inoue Yasunao,Omodani Tomoki,Shiratake Ryotaro,Sato Fuminori

Publisher

Elsevier BV

Subject

Inorganic Chemistry,Organic Chemistry,Physical and Theoretical Chemistry,Catalysis

Reference16 articles.

1. Development of a highly water-soluble peptide-based human neutrophil elastase inhibitor; AE-3763 for treatment of acute organ injury

2. Sato, F.; Inoue, Y.; Omodani, T.; Shiratake, R.; Honda, S.; Komiya, M.; Takemura, T. Int. Pat. Appl. WO 2000/052032, 2000.

3. Imidazo[1,2-a]piperazines as mechanistic inhibitors of serine proteinases

4. elastase inhibitors containing conformationally restricted lactams as P3-P2 dipeptide replacements

5. Inhibition of Human Neutrophil Elastase with Peptidyl Electrophilic Ketones. 2. Orally Active PG-Val-Pro-Val Pentafluoroethyl Ketones

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