Selectively targeting the dimerization interface of human androgen receptor with small-molecules to treat castration-resistant prostate cancer
Author:
Funder
Canadian Institutes of Health Research (CIHR
Prostate Cancer Canada-Translational Acceleration
Terry Fox New Frontiers Program
Publisher
Elsevier BV
Subject
Cancer Research,Oncology
Reference44 articles.
1. Androgen action and metabolism in prostate cancer;Green;Mol. Cell. Endocrinol.,2012
2. Targeting alternative sites on the androgen receptor to treat castration-resistant prostate cancer;Lallous;Int. J. Mol. Sci.,2013
3. Domains of the human androgen receptor involved in steroid binding, transcriptional activation, and subcellular localization;Jenster;Mol. Endocrinol.,1991
4. Treatment options in castration-resistant prostate cancer: current therapies and emerging docetaxel-based regimens;Saad;Urol. Oncol.,2014
5. Structural basis for accommodation of nonsteroidal ligands in the androgen receptor;Bohl;J. Biol. Chem.,2005
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