An experimental method for the determination of enzyme-competitive inhibitor dissociation constants from displacement curves: Application to human renin using fluorescence energy transfer to a synthetic dansylated inhibitor peptide-Reference-Cited by-同舟云学术

An experimental method for the determination of enzyme-competitive inhibitor dissociation constants from displacement curves: Application to human renin using fluorescence energy transfer to a synthetic dansylated inhibitor peptide

Published:1989-08 Issue:1 Volume:181 Page:172-181
ISSN:0003-2697
Container-title:Analytical Biochemistry
language:en
Short-container-title:Analytical Biochemistry

Author:

Epps Dennis E.,Schostarez Heinrich,Argoudelis Christine V.,Poorman Roger,Hinzmann Jessica,Sawyer Tomi K.,Mandel Frederic

Publisher

Elsevier BV

Subject

Cell Biology,Molecular Biology,Biochemistry,Biophysics

Reference13 articles.

1. Interrelations between various blood pressure regulatory systems and the mosaic theory of hypertension

2. Potent new inhibitors of human renin

3. Design, structure-activity, and molecular modeling studies of potent renin inhibitory peptides having N-terminal Nin-For-Trp (Ftr): angiotensinogen congeners modified by P1-P1' Phe-Phe, Sta, Leu.psi.[CH(OH)CH2]Val or Leu.psi.[CH2NH]Val substitutions

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