Structural characterization of inhibitor complexes with checkpoint kinase 2 (Chk2), a drug target for cancer therapy-Reference-Cited by-同舟云学术

Structural characterization of inhibitor complexes with checkpoint kinase 2 (Chk2), a drug target for cancer therapy

Published:2011-12 Issue:3 Volume:176 Page:292-301
ISSN:1047-8477
Container-title:Journal of Structural Biology
language:en
Short-container-title:Journal of Structural Biology

Author:

Lountos George T.,Jobson Andrew G.,Tropea Joseph E.,Self Christopher R.,Zhang Guangtao,Pommier Yves,Shoemaker Robert H.,Waugh David S.

Publisher

Elsevier BV

Subject

Structural Biology

Reference65 articles.

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3. CCT241533 is a potent and selective inhibitor of CHK2 that potentiates the cytotoxicity of PARP inhibitors;Anderson;Cancer Res.,2011

4. CHK2 kinase: cancer susceptibility and cancer therapy – two sides of the same coin?;Antoni;Nat. Rev. Cancer,2007

5. Checkpoint kinase inhibitors: SAR and radioprotective properties of a series of 2-arylbenzimidazoles;Arienti;J. Med. Chem.,2005

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