On the fundamental difference in the thermodynamics of agonist and antagonist interactions with β-adrenergic receptors and the mechanism of entropy-driven binding-Reference-Cited by-同舟云学术

On the fundamental difference in the thermodynamics of agonist and antagonist interactions with β-adrenergic receptors and the mechanism of entropy-driven binding

Published:1990-08 Issue:4 Volume:40 Page:663-669
ISSN:0006-2952
Container-title:Biochemical Pharmacology
language:en
Short-container-title:Biochemical Pharmacology

Author:

Miklavc Adolf,Kocjan Darko,Mavri Jonez,Koller Jože,Hadži Dušan

Publisher

Elsevier BV

Subject

Pharmacology,Biochemistry

Reference44 articles.

1. Fundamental difference between the molecular interactions of agonists and antagonists with the β-adrenergic receptor;Weiland;Nature,1979

2. Influence of temperature on the sensivitity of the β-receptors and the contractility of guinea-pig atrium;Reinhardt;Naunyn-Schmiedebergs Arch Pharmacol,1972

3. Temperature dependent supersensitivity of isolated atria to catecholamines;Wöppel;Eur J Pharmacol,1973

4. Studies on the temperature-dependent sensitivity of mouse atria to adrenergic drugs;Mun̄oz-Ramirez;Eur J Pharmacol,1975

5. Agonist-specific alterations in receptor binding affinity associated with solubilization of turkey erythrocyte membrane beta-adrenergic receptors;Pike;Mol Pharmacol,1978

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