Synthesis of propynyloxy substituted some novel aurones as potent cathepsin B inhibitors
Author:
Funder
Haryana State Council for Science and Technology
Publisher
Elsevier BV
Subject
General Chemistry
Reference51 articles.
1. Cathepsin B is a new drug target for traumatic brain injury therapeutics: evidence for E64d as a promising lead drug candidate;Hook;Front. Neurol.,2015
2. Cathepsin B activates human trypsinogen 1 but not proelastase 2 or procarboxypeptidase B;Lindkvist;Pancreatology,2006
3. Microglial cathepsin B as a key driver of inflammatory brain diseases and brain aging;Nakanishi;Neural Regen. Res.,2020
4. Overexpression of cathepsin B in gastric cancer identified by proteome analysis;Ebert;Proteomics,2005
5. Cathepsin B promotes both motility and invasiveness of oral carcinoma cells;Wickramasinghe;Arch. Biochem. Biophys.,2005
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