Asymmetric synthesis of β-aryl-β-trifluoromethyl-β-aminoarones via Mannich-type reactions of ketone enolates with chiral aryl CF3-substituted N-tert-butanesulfinyl ketimines
Author:
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Reference40 articles.
1. Modern Variants of the Mannich Reaction
2. Evolution of the Vinylogous Mannich Reaction as a Key Construction for Alkaloid Synthesis
3. Simple and Efficient Access to N-Tosyl β-Amino Ketones and Their Conversion into 2,4-Disubstituted Azetidines
4. Total synthesis of (5R,6R,8R,9S)-(−)-5,9Z-indolizidine 221T using sulfinimine-derived N-sulfinyl β-amino ketones
5. Asymmetric Synthesis of Substituted Tropinones Using the Intramolecular Mannich Cyclization Reaction and Acyclic N-Sulfinyl β-Amino Ketone Ketals
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