Cereblon neo-substrate binding mimics the recognition of the cyclic imide degron
Author:
Funder
Max-Planck-Gesellschaft
Paul Scherrer Institut
Publisher
Elsevier BV
Subject
Cell Biology,Molecular Biology,Biochemistry,Biophysics
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1. Revisiting the antiangiogenic mechanisms of fluorinated thalidomide derivatives;Bioorganic & Medicinal Chemistry Letters;2024-09
2. IKZF2 Degradation: It′s Time to Take into Account it When Designing Cereblon‐Based PROTACs;ChemBioChem;2024-07-11
3. Strengthening Molecular Glues: Design Strategies for Improving Thalidomide Analogs as Cereblon Effectors and Anticancer Agents;Drug Discovery Today;2024-06
4. Targeted protein degradation: from mechanisms to clinic;Nature Reviews Molecular Cell Biology;2024-04-29
5. Discovery and characterization of potent spiro-isoxazole-based cereblon ligands with a novel binding mode;European Journal of Medicinal Chemistry;2024-04
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