The development of A-ring modified analogues of oestrone-3-O-sulphamate as potent steroid sulphatase inhibitors with reduced oestrogenicity-Reference-Cited by-同舟云学术

The development of A-ring modified analogues of oestrone-3-O-sulphamate as potent steroid sulphatase inhibitors with reduced oestrogenicity

Published:1998-03 Issue:5-6 Volume:64 Page:269-275
ISSN:0960-0760
Container-title:The Journal of Steroid Biochemistry and Molecular Biology
language:en
Short-container-title:The Journal of Steroid Biochemistry and Molecular Biology

Author:

Purohit A.,Vernon K.A.,Wagenaar Hummelinck A.E.,Woo L.W.L.,Hejaz H.A.M.,Potter B.V.L.,Reed M.J.

Publisher

Elsevier BV

Subject

Cell Biology,Clinical Biochemistry,Endocrinology,Molecular Biology,Molecular Medicine,Biochemistry,Endocrinology, Diabetes and Metabolism

Reference27 articles.

1. Importance of estrogen sulfates in breast cancer;Pasqualini;J. Steroid Biochem. Molec. Biol.,1989

2. Estrone sulfate stimulates growth of nitrosomethylurea induced breast carcinoma in vivo in the rat;Santner;Int. J. Cancer,1990

3. Concentrations of estrone, estradiol and estrone sulfate and evaluation of sulfatase and aromatase activities in pre- and postmenopausal breast cancer patients;Pasqualini;J. Clin. Endocr. Metab.,1996

4. In situ estrogen production via estrone sulfatase pathway in breast tumors: Relative importance vs aromatase pathway;Santner;J. Clin. Endocrinol. Metab.,1984

5. Stimulation of cell proliferation and estrogenic response by adrenal C19-delta-5-steroids in ZR-75-1 human breast cancer cell line;Poulin;Cancer Res.,1986

Cited by 96 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Potent Dual Inhibitors of Steroid Sulfatase and 17β-Hydroxysteroid Dehydrogenase Type 1 with a Suitable Pharmacokinetic Profile for In Vivo Proof-of-Principle Studies in an Endometriosis Mouse Model;Journal of Medicinal Chemistry;2023-06-27

2. Dual Targeting of Steroid Sulfatase and 17β-Hydroxysteroid Dehydrogenase Type 1 by a Novel Drug-Prodrug Approach: A Potential Therapeutic Option for the Treatment of Endometriosis;Journal of Medicinal Chemistry;2022-08-22

3. Steroid Sulphatase and Its Inhibitors: Past, Present and Future;Molecules;2021-05-11

4. Recent Developments in Coumarin Derivatives for Breast Cancer Therapy;International Journal of Advanced Research in Science, Communication and Technology;2020-12-11

5. Direct quantification of anorethidrani disuccinate and determination of sterol metabolites by chemical derivatization combined with LC-MS/MS: Application to a Phase I pharmacokinetic study in humans;Journal of Chromatography B;2020-11