In vitro–in vivo correlation for wet-milled tablet of poorly water-soluble cilostazol

Author:

Jinno Jun-ichi,Kamada Naoki,Miyake Masateru,Yamada Keigo,Mukai Tadashi,Odomi Masaaki,Toguchi Hajime,Liversidge Gary G.,Higaki Kazutaka,Kimura Toshikiro

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference39 articles.

1. Poorly aqueous solubility: an industry wide problem in drug discovery;Lipinski;Am. Pharm. Rev.,2002

2. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings;Lipinski;Adv. Drug Deliv. Rev.,2001

3. Drug-like properties and the causes of poor solubility and poor permeability;Lipinski;J. Pharmacol. Toxicol. Methods,2000

4. Drug delivery strategies for poorly water-soluble drugs;Fahr;Expert Opin. Drug Deliv.,2007

5. Solid dispersions of poorly water-soluble drugs: early promises, subsequent problems, and recent breakthroughs;Serajuddin;J. Pharm. Sci.,1999

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