Kinetic mechanism of dopamine transporter interaction with 1-(2-(bis-(4-fluorophenyl)methoxy)ethyl)-4-(3-phenylpropyl)piperazine (GBR 12909)
Author:
Publisher
Elsevier BV
Subject
Cell Biology,Cellular and Molecular Neuroscience
Reference15 articles.
1. High affinity [3H]GBR 12783 binding to a specific site associated with the neuronal dopamine uptake complex in the central nervous system;Bonnet;Eur. J. Pharmacol.,1986
2. Relationship between inhibition constant (Ki) and concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic-reaction;Cheng;Biochem. Pharmacol.,1973
3. Evidence for the sequential formation of two complexes between an uptake inhibitor, GBR 12783 [1-[2-(diphenylmethoxy)ethyl]-4-(3-phenyl-2-propenyl)piperazine], and the neuronal transporter of dopamine;Do-Rego;J. Neurochem.,1999
4. Synthesis and ligand binding of nortropane derivatives: N-substituted-2β-carbomethoxy-3β-(4′-iodophenyl) nortropane and N-(3-iodoprop-(2E)-enyl)-2β-carbomethoxy-3β-(3′,4′-disubstitutedphenyl) nortropane. New high-affinity and selective compounds for the dopamine transporter;Emond;J. Med. Chem.,1997
5. PET study of the pre- and post-synaptic dopaminergic markers for the neurodegenerative process in Huntington’s disease;Ginovart;Brain,1997
Cited by 6 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. The influence of acute dopamine transporter inhibition on manic-, depressive-like phenotypes, and brain oxidative status in adult zebrafish;Progress in Neuro-Psychopharmacology and Biological Psychiatry;2024-04
2. Daily Monitoring of Dopamine Efflux Reveals a Short-Lasting Occlusion of the Dopamine Agonist Properties of d-Amphetamine by Dopamine Transporter Blockers GBR 12909 and Methylphenidate;ACS Chemical Neuroscience;2013-05-03
3. Latest Advancements on Serotonin and Dopamine Transporters in Lymphocytes;Mini-Reviews in Medicinal Chemistry;2010-01-01
4. A new model of the disrupted latent inhibition in C57BL/6J mice after bupropion treatment;Psychopharmacology;2009-12-16
5. Behavioural characterisation of the effects of acute and repeated administration of GBR 12909 in rats: Further evaluation of a potential model of ADHD;Neuropharmacology;2009-12
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3