The isoquinoline PRL-295 increases the thermostability of Keap1 and disrupts its interaction with Nrf2-Reference-Cited by-同舟云学术

The isoquinoline PRL-295 increases the thermostability of Keap1 and disrupts its interaction with Nrf2

Published:2022-01 Issue:1 Volume:25 Page:103703
ISSN:2589-0042
Container-title:iScience
language:en
Short-container-title:iScience

Author:

Dayalan Naidu Sharadha,Suzuki Takafumi,Dikovskaya Dina,Knatko Elena V.,Higgins Maureen,Sato Miu,Novak Miroslav,Villegas José A.,Moore Terry W.,Yamamoto Masayuki,Dinkova-Kostova Albena T.

Publisher

Elsevier BV

Subject

Multidisciplinary

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4. Design, synthesis, and evaluation of triazole derivatives that induce Nrf2 dependent gene products and inhibit the Keap1-Nrf2 protein-protein interaction;Bertrand;J. Med. Chem.,2015

5. Can activation of NRF2 Be a strategy COVID-19?;Cuadrado;Trends Pharmacol. Sci.,2020

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