Voltage-Gated Sodium Channel Drug Discovery Technologies and Challenges
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InTech
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http://www.intechopen.com/download/pdf/63174
Reference17 articles.
1. Chernov-Rogan T, Li T, Lu G, Verschoof H, Khakh K, et al. Mechanism-specific assay design facilitates the discovery of Nav1.7-selective inhibitors. Proceedings of the National Academy of Sciences of the United States of America. 2018;115:E792-E801. DOI: 10.1073/pnas.1713701115
2. Pellecchia M, Bertini I, Cowburn D, Dalvit C, Giralt E, et al. Perspectives on NMR in drug discovery: A technique comes of age. Nature Reviews Drug Discovery. 2008;7:738-745. DOI: 10.1038/nrd2606
3. Finley M, Cassaday J, Kreamer T, Li X, Solly K, et al. Kinetic analysis of membrane potential dye response to Nav1.7 channel activation identifies antagonists with pharmacological selectivity against Nav1.5. Journal of Biomolecular Screening. 2016;21:480-489. DOI: 10.1177/1087057116629669
4. Liu CJ, Priest BT, Bugianesi RM, Dulski PM, Felix JP, et al. A high-capacity membrane potential FRET-based assay for Nav1.8 channels. Assay and Drug Development Technologies. 2006;4:37-48. DOI: 10.1089/adt.2006.4.37
5. Fitch RW, Daly JW. Phosphorimaging detection and quantitation for isotopic ion flux assays. Analytical Biochemistry. 2005;342:260-270. DOI: 10.1016/j.ab.2005.04.041
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