Author:
Holan George,Virgona Christopher,Watson Keith G.
Abstract
5-Chloro-1-methyl-1,2-dihydro-3H-1,2,4-triazol-3-one
(12) and
N-isopropyl-2-methyl-5-oxo-2,5-dihydro-1H1,2,4triazole3-sulfonamide
(14) have been prepared from 1-methyl-5-thioxo-1,2,4-triazolidin-3-one (7) and
converted into the methanesulfonate esters (15) and (16). The
anti-acetylcholinesterase and insecticidal activities of (15) and (16) have
been compared with those of the known
5-isobutylthio-1-methyl-1H-1,2,4-triazol-3-yl
methanesulfontate (4).
Cited by
6 articles.
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2. Some urea and thiourea derivatives bearing 1,2,4-triazole ring and their anti-acetylcholinesterase activities;Journal of Marmara University Institute of Health Sciences;2014
3. Synthesis, Antifungal Activity, and Docking Study of Some New 1,2,4-triazole Analogs;Chemical Biology & Drug Design;2011-09-26
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