Abstract
Syntheses are described for
several 4-(1',2',4'-triazol-3'yl)pyridines,
3-and 4-(1',3',4'-thiadiazol-2'-yl)-pyridines,
3- and 4-(1',3',4'-oxadiazol-2'-yl)pyridines, 5-(1',3',4'-thiadiazol-2'-yl)pyrimidines
and 5-(1',3',4'-oxadiazol-2'-yl)pyrimidines,
all provided
with a β-dimethylaminoethylthio side chain at the
5-position of the five-membered ring. The activities of these compounds as
amplifiers of phleomycin-G against an in vitro culture of Escherichia coli B are tabulated and discussed.
Cited by
14 articles.
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