The macrolide drug erythromycin does not protect the hERG channel from inhibition by thioridazine and terfenadine-Reference-Cited by-同舟云学术

The macrolide drug erythromycin does not protect the hERG channel from inhibition by thioridazine and terfenadine

Published:2020-03 Issue:5 Volume:8 Page:
ISSN:2051-817X
Container-title:Physiological Reports
language:en
Short-container-title:Physiol Rep

Author:

El Harchi Aziza¹^ORCID,Butler Andrew S.¹^ORCID,Zhang Yihong¹,Dempsey Christopher E.²^ORCID,Hancox Jules C.¹^ORCID

Affiliation:

1. School of Physiology and Pharmacology and Neuroscience Biomedical Sciences Building The University of Bristol University Walk Bristol UK

2. School of Biochemistry Biomedical Sciences Building The University of Bristol University Walk Bristol UK

Funder

Heart Research UK

Publisher

Wiley

Subject

Physiology (medical),Physiology

Link

https://onlinelibrary.wiley.com/doi/pdf/10.14814/phy2.14385

Reference49 articles.

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3. Theoretical Basis, Experimental Design, and Computerized Simulation of Synergism and Antagonism in Drug Combination Studies

4. Loratadine blockade of K+ channels in human heart: Comparison with terfenadine under physiological conditions;Crumb W. J.;Journal of Pharmacology and Experimental Therapeutics,2000

5. Allosteric effects of erythromycin pretreatment on thioridazine block of hERG potassium channels

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