Synthesis and Antibacterial Activity of Novel Vanillic Acid Hybrid Derivatives [Part II]-Reference-Cited by-同舟云学术

Synthesis and Antibacterial Activity of Novel Vanillic Acid Hybrid Derivatives [Part II]

Published:2018-12-03 Issue: Volume: Page:219-223
ISSN:2395-602X
Container-title:International Journal of Scientific Research in Science and Technology
language:en
Short-container-title:IJSRST

Author:

S. Satpute Maruti¹,D. Gangan Vijay²,Shastri Indu¹

Affiliation:

1. Departement of Chemistry, R. D. National College and W. A. Science College, Linking Road, Bandra, Mumbai, Maharastra, India

2. Department of Chemistry, Loba R & D Centre, Loba Chemie Pvt. Ltd., Plot No. D - 22, Tarapur MIDC, Boisar, Palghar, Maharastra, India

Abstract

Vanillic acid (4-hydroxy-3-methoxybenzoic acid) is a dihydroxybenzoic acid derivative used as a flavoring agent. It is used in the synthesis of various active pharmaceutical ingredients such as Etamivan, Modecainide, Brovanexine, Vanitiolide, Vanyldisulfamide etc. In this paper, novel ester / hybrid derivatives of vanillic acid were synthesized and tested for potential antibacterial activity. This combinatorial synthesis of novel vanillic ester / hybrid derivatives can be a useful approach to generate potent chemotherapeutic agents in developing new drug candidates.

Publisher

Technoscience Academy

Subject

General Medicine

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