Measurement of Tafenoquine (WR 238605) in Human Plasma and Venous and Capillary Blood by High-Pressure Liquid Chromatography
Author:
Publisher
Ovid Technologies (Wolters Kluwer Health)
Subject
Pharmacology (medical),Pharmacology
Reference6 articles.
1. Prophylaxis of Plasmodium falciparum Infection in a Human Challenge Model with WR 238605, a New 8-Aminoquinoline Antimalarial
2. First-time-in-humans safety and pharmacokinetics of WR 238605, a new antimalarial.
3. Rapid and sensitive quantitative analysis of the new antimalarial N4-[2,6-dimethoxy-4-methyl-5-[(3-trifluoromethyl)phenoxy]-8-quinolinyl]-1,4-pentanediamine in plasma by liquid chromatography and electrochemical detection
4. Quantification of the individual enantiomer plasma concentrations of the candidate antimalarial agent N4-[2,6-dimethoxy-4-methyl-5-[(3-trifluoromethyl)phenoxyl]-8-quinolinyl]-1,4-pentanediamine (WR 238,605)
5. High-performance liquid chromatographic assay for the simultaneous monitoring of mefloquine and its acid metabolite in biological samples using protein precipitation and ion-pair extraction
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1. Cytochrome P450 2D6 profiles and anti-relapse efficacy of tafenoquine against Plasmodium vivax in Australian Defence Force personnel;Antimicrobial Agents and Chemotherapy;2023-12-14
2. Quantification of Tafenoquine and 5,6-Orthoquinone Tafenoquine by UHPLC-MS/MS in Blood, Plasma, and Urine, and Application to a Pharmacokinetic Study;Molecules;2022-11-24
3. Determination of tafenoquine in human plasma by dispersive liquid‐liquid microextraction;SEPARATION SCIENCE PLUS;2020-01-20
4. Dried Blood Spots for Global Health Diagnostics and Surveillance: Opportunities and Challenges;The American Journal of Tropical Medicine and Hygiene;2018-08-02
5. Differential Cytochrome P450 2D Metabolism Alters Tafenoquine Pharmacokinetics;Antimicrobial Agents and Chemotherapy;2015-04-13
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