Chimeric α 2 -,β 2 -Adrenergic Receptors: Delineation of Domains Involved in Effector Coupling and Ligand Binding Specificity

Author:

Kobilka Brian K.1,Kobilka Tong Sun1,Daniel Kiefer1,Regan John W.1,Caron Marc G.1,Lefkowitz Robert J.1

Affiliation:

1. Howard Hughes Medical Institute, Department of Medicine, Duke University Medical Center, Durham, NC 27710.

Publisher

American Association for the Advancement of Science (AAAS)

Subject

Multidisciplinary

Reference17 articles.

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2. DELEAN, A, AM J PHYSIOL 235: 97 (1978).

3. DELEAN, A, VALIDATION AND STATISTICAL-ANALYSIS OF A COMPUTER MODELING METHOD FOR QUANTITATIVE-ANALYSIS OF RADIOLIGAND BINDING DATA FOR MIXTURES OF PHARMACOLOGICAL RECEPTOR SUBTYPES, MOLECULAR PHARMACOLOGY 21: 5 (1982).

4. DIXON, RAF, STRUCTURAL FEATURES REQUIRED FOR LIGAND-BINDING TO THE BETA-ADRENERGIC-RECEPTOR, EMBO JOURNAL 6: 3269 (1987).

5. Ligand binding to the β-adrenergic receptor involves its rhodopsin-like core

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