NUCKS1 promotes invasion and metastasis of colorectal cancer by stabilizing HDAC2 and activating AKT

Author:

Song Yang,Zhu Liaoliao,Zhao ting,Su Haichuan1ORCID,Li Junqiang,Shen jing,Zhang liang,Chen jun

Affiliation:

1. Tangdu Hospital, Air Force Medical University

Abstract

Abstract

Nuclear ubiquitous casein and cyclin-dependent kinase substrate 1 (NUCKS1) functions as an oncogene in colorectal cancer (CRC), promotes the progression of CRC, and is associated with poor prognosis in patients. Studies have found that NUCKS1 promotes tumor cell metastasis, yet its role in CRC invasion and metastasis remains unclear. To investigate this, transwell migration and invasion assay, wound healing assay, and immunofluorescence assay were performed in vitro. Additionally, label-free protein quantification, coimmunoprecipitation (Co-IP), q-PCR, and Western blotting were utilized to analyze NUCKS1's molecular mechanisms in CRC. In vivo, CRC cells were injected into the tail vein to examine NUCKS1's impact on lung and liver metastasis in mice, with hematoxylin-eosin (HE) staining used to evaluate metastatic lesion sizes. Results indicated higher NUCKS1 expression in metastatic CRC compared to non-metastatic samples. Knockdown of NUCKS1 in vitro inhibited CRC invasion and metastasis. Moreover, NUCKS1 was initially found to upregulate HDAC2 expression by inhibiting the lysosomal pathway, activating AKT, and thus promoting CRC invasion and metastasis. In vivo, overexpression of NUCKS1-induced lung and liver metastasis was suppressed by HDAC2 knockdown or intraperitoneal administration of the HDAC2 inhibitor Santacruzamate A. These findings suggest that NUCKS1 contributes to CRC invasion and metastasis by stabilizing HDAC2 and activating AKT, highlighting NUCKS1 and HDAC2 as potential therapeutic targets for CRC.

Publisher

Springer Science and Business Media LLC

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3