An 19f Nmr Fragment-Based Approach for the Discovery and Development of Brca2-Rad51 Inhibitors to Pursuit Synthetic Lethality in Combination with Parp Inhibition in Pancreatic Cancer

Author:

Myers Samuel,Poppi Laura,Rinaldi Francesco,Veronesi Marina,Ciamarone Andrea,Previtali Viola,Bagnolini Greta,Schipani Fabrizio,Ortega Martínez Jose Antonio,Girotto Stefania,Di Stefano Giuseppina,Farabegoli Fulvia,Walsh Naomi,De Franco Francesca,Roberti Marinella,Cavalli Andrea

Publisher

Elsevier BV

Reference58 articles.

1. DNA Damage and Its Role in Cancer Therapeutics;J Moon;Int J Mol Sci

2. DNA damage repair: historical perspectives, mechanistic pathways and clinical translation for targeted cancer therapy;R Huang;Signal Transduction and Targeted Therapy

3. Population Frequency of Germline BRCA1/2 Mutations;K N Maxwell;Journal of Clinical Oncology,2016

4. Synthetic Lethality in Pancreatic Cancer: Discovery of a New RAD51-BRCA2 Small Molecule Disruptor That Inhibits Homologous Recombination and Synergizes with Olaparib;G Bagnolini;Journal of Medicinal Chemistry,2020

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