Incorporation of the Time-Varying Postprandial Increase in Splanchnic Blood Flow into a PBPK Model to Predict the Effect of Food on the Pharmacokinetics of Orally Administered High-Extraction Drugs-Reference-Cited by-同舟云学术

Incorporation of the Time-Varying Postprandial Increase in Splanchnic Blood Flow into a PBPK Model to Predict the Effect of Food on the Pharmacokinetics of Orally Administered High-Extraction Drugs

Published:2017-05-19 Issue:4 Volume:19 Page:1205-1217
ISSN:1550-7416
Container-title:The AAPS Journal
language:en
Short-container-title:AAPS J

Author:

Rose Rachel H.,Turner David B.,Neuhoff Sibylle,Jamei Masoud

Publisher

Springer Science and Business Media LLC

Subject

Pharmaceutical Science

Link

http://link.springer.com/article/10.1208/s12248-017-0099-z/fulltext.html

Reference76 articles.

1. Welling PG. Effects of food on drug absorption. Annu Rev Nutr. 1996;16:383–415.

2. FDA. Guidance for industry: food-effect bioavailability and fed bioequivalence studies. Rockville, MD: Food and Drug Administration; 2002.

3. Andreas CJ, Pepin X, Markopoulos C, Vertzoni M, Reppas C, Dressman JB. Mechanistic investigation of the negative food effect of modified release zolpidem. Eur J Pharm Sci. 2017;102:284–98.

4. Cristofoletti R, Patel N, Dressman JB. Differences in food effects for 2 weak bases with similar BCS drug-related properties: what is happening in the intestinal lumen? J Pharm Sci. 2016;105(9):2712–22.

5. Heimbach T, Xia B, Lin TH, He H. Case studies for practical food effect assessments across BCS/BDDCS class compounds using in silico, in vitro, and preclinical in vivo data. AAPS J. 2013;15(1):143–58.

Cited by 24 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. A guide to developing population files for physiologically‐based pharmacokinetic modeling in the Simcyp Simulator;CPT: Pharmacometrics & Systems Pharmacology;2024-07-18

2. Analysis of the interplay of physiological response to food intake and drug properties in food-drug interactions;Drug Metabolism and Pharmacokinetics;2023-12

3. Application of physiologically based pharmacokinetics modeling in the research of small-molecule targeted anti-cancer drugs;Cancer Chemotherapy and Pharmacology;2023-07-19

4. A Physiologically-Based Pharmacokinetic Model for Cannabidiol in Healthy Adults, Hepatically-Impaired Adults, and Children;Drug Metabolism and Disposition;2023-03-27

5. Assessment of food effects during clinical development;International Journal of Pharmaceutics;2023-03