Mathematical Models to Explore Potential Effects of Supersaturation and Precipitation on Oral Bioavailability of Poorly Soluble Drugs
Author:
Publisher
Springer Science and Business Media LLC
Subject
Pharmaceutical Science
Link
http://link.springer.com/content/pdf/10.1208/s12248-015-9748-2.pdf
Reference51 articles.
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3. Murdande SB, Pikal MJ, Shanker RM, Bogner RH. Solubility advantage of amorphous pharmaceuticals, part 3: is maximum solubility advantage experimentally attainable and sustainable? J Pharm Sci. 2011;100(10):4349–56.
4. Brouwers J, Brewster ME, Augustijns P. Supersaturating drug delivery systems: the answers to solubility-limited bioavailability? J Pharm Sci. 2008;98(8):2549–72.
5. Greco K, Bogner R. Solution-mediated phase transformation: significance during dissolution and implications for bioavailability. J Pharm Sci. 2012;101(9):2996–3018.
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