Evaluation of Tadalafil Nanosuspensions and Their PEG Solid Dispersion Matrices for Enhancing Its Dissolution Properties

Author:

Obeidat Wasfy M.,Sallam Al-Sayed A.

Publisher

Springer Science and Business Media LLC

Subject

Drug Discovery,Pharmaceutical Science,Agronomy and Crop Science,Ecology,Aquatic Science,General Medicine,Ecology, Evolution, Behavior and Systematics

Reference38 articles.

1. Lomabardino JG, Lowe III JA. A guide to drug discovery: the role of the medicinal chemist in drug discovery—then and now. Nat Rev Drug Discov. 2004;3:853–62.

2. Thomas R. Solubility enhancement with BASF pharma polymers. Lampertheim: BASF SE Pharma Ingredients & Services; 2011.

3. Keck CM, Muller RH. Drug nanocrystals of poorly soluble drugs produced by high pressure homogenisation. Eur J Pharm Biopharm. 2006;62:3–16.

4. Lipinski C. Poor aqueous solubility—an industry wide problem in drug discovery. Am Pharm Rev. 2002;5:82–5.

5. Patro S, Himasankar K, Choudhury AA, Rao MEB. Effect of some hydrophilic polymers on dissolution rate of roxitromycin. Indian J Pharm Sci. 2005;67:334–41.

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