Turning a protein kinase on or off from a single allosteric site via disulfide trapping
Author:
Publisher
Proceedings of the National Academy of Sciences
Subject
Multidisciplinary
Reference29 articles.
1. Site-directed ligand discovery
2. Tethering: Fragment-Based Drug Discovery
3. Discovery of an allosteric site in the caspases
4. Disulfide trapping to localize small-molecule agonists and antagonists for a G protein-coupled receptor
5. Site-specific Disulfide Capture of Agonist and Antagonist Peptides on the C5a Receptor
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