A small-molecule mimic of a peptide docking motif inhibits the protein kinase PDK1-Reference-Cited by-同舟云学术

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A small-molecule mimic of a peptide docking motif inhibits the protein kinase PDK1

Published:2014-12-17 Issue:52 Volume:111 Page:18590-18595
ISSN:0027-8424
Container-title:Proceedings of the National Academy of Sciences
language:en
Short-container-title:Proc Natl Acad Sci USA

Author:

Rettenmaier T. Justin,Sadowsky Jack D.,Thomsen Nathan D.,Chen Steven C.,Doak Allison K.,Arkin Michelle R.,Wells James A.

Funder

HHS | National Institutes of Health (NIH)

HHS | NIH | National Cancer Institute (NCI)

Tobacco-Related Disease Research Program (TRDRP)

Damon Runyon Cancer Research Foundation (Damon Runyon)

Publisher

Proceedings of the National Academy of Sciences

Subject

Multidisciplinary

Reference34 articles.

1. Strategies for the Selective Regulation of Kinases with Allosteric Modulators: Exploiting Exclusive Structural Features

2. Catalytic Control in the EGF Receptor and Its Connection to General Kinase Regulatory Mechanisms

3. The nuts and bolts of AGC protein kinases

4. Selective 3-Phosphoinositide-Dependent Kinase 1 (PDK1) Inhibitors: Dissecting the Function and Pharmacology of PDK1

5. Identification of a pocket in the PDK1 kinase domain that interacts with PIF and the C-terminal residues of PKA

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1. Conserved regulatory motifs in the juxtamembrane domain and kinase N-lobe revealed through deep mutational scanning of the MET receptor tyrosine kinase domain;eLife;2024-09-13

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3. Conserved regulatory motifs in the juxtamembrane domain and kinase N-lobe revealed through deep mutational scanning of the MET receptor tyrosine kinase domain;2024-06-26

4. Targeting the PDK/PDH axis to reverse metabolic abnormalities by structure-based virtual screening with in vitro and in vivo experiments;International Journal of Biological Macromolecules;2024-03

5. A virtual library of small molecules mimicking dipeptides;Archiv der Pharmazie;2024-02-08

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