Small molecule inhibitors of mesotrypsin from a structure-based docking screen
Author:
Funder
National Cancer Institute
Publisher
Public Library of Science (PLoS)
Subject
Multidisciplinary
Reference46 articles.
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2. Crystal structure reveals basis for the inhibitor resistance of human brain trypsin;G Katona;J Mol Biol,2002
3. Human mesotrypsin is a unique digestive protease specialized for the degradation of trypsin inhibitors;R Szmola;J Biol Chem,2003
4. Activity of recombinant trypsin isoforms on human proteinase-activated receptors (par): Mesotrypsin cannot activate epithelial par-1, -2, but weakly activates brain par-1;Z Grishina;Br J Pharmacol,2005
5. Trypsin IV or mesotrypsin and p23 cleave protease-activated receptors 1 and 2 to induce inflammation and hyperalgesia;W Knecht;J Biol Chem,2007
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